RT Journal Article T1 THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors. A1 Alexander, Stephen Ph A1 Christopoulos, Arthur A1 Davenport, Anthony P A1 Kelly, Eamonn A1 Mathie, Alistair A1 Peters, John A A1 Veale, Emma L A1 Armstrong, Jane F A1 Faccenda, Elena A1 Harding, Simon D A1 Pawson, Adam J A1 Southan, Christopher A1 Davies, Jamie A A1 Abbracchio, Maria Pia A1 Alexander, Wayne A1 Al-Hosaini, Khaled A1 Bäck, Magnus A1 Barnes, Nicholas M A1 Bathgate, Ross A1 Beaulieu, Jean-Martin A1 Bernstein, Kenneth E A1 Bettler, Bernhard A1 Birdsall, Nigel J M A1 Blaho, Victoria A1 Boulay, Francois A1 Bousquet, Corinne A1 Bräuner-Osborne, Hans A1 Burnstock, Geoffrey A1 Caló, Girolamo A1 Castaño, Justo P A1 Catt, Kevin J A1 Ceruti, Stefania A1 Chazot, Paul A1 Chiang, Nan A1 Chini, Bice A1 Chun, Jerold A1 Cianciulli, Antonia A1 Civelli, Olivier A1 Clapp, Lucie H A1 Couture, Réjean A1 Csaba, Zsolt A1 Dahlgren, Claes A1 Dent, Gordon A1 Singh, Khuraijam Dhanachandra A1 Douglas, Steven D A1 Dournaud, Pascal A1 Eguchi, Satoru A1 Escher, Emanuel A1 Filardo, Edward J A1 Fong, Tung A1 Fumagalli, Marta A1 Gainetdinov, Raul R A1 Gasparo, Marc de A1 Gerard, Craig A1 Gershengorn, Marvin A1 Gobeil, Fernand A1 Goodfriend, Theodore L A1 Goudet, Cyril A1 Gregory, Karen J A1 Gundlach, Andrew L A1 Hamann, Jörg A1 Hanson, Julien A1 Hauger, Richard L A1 Hay, Debbie L A1 Heinemann, Akos A1 Hollenberg, Morley D A1 Holliday, Nicholas D A1 Horiuchi, Mastgugu A1 Hoyer, Daniel A1 Hunyady, László A1 Husain, Ahsan A1 IJzerman, Adriaan P A1 Inagami, Tadashi A1 Jacobson, Kenneth A A1 Jensen, Robert T A1 Jockers, Ralf A1 Jonnalagadda, Deepa A1 Karnik, Sadashiva A1 Kaupmann, Klemens A1 Kemp, Jacqueline A1 Kennedy, Charles A1 Kihara, Yasuyuki A1 Kitazawa, Takio A1 Kozielewicz, Pawel A1 Kreienkamp, Hans-Jürgen A1 Kukkonen, Jyrki P A1 Langenhan, Tobias A1 Leach, Katie A1 Lecca, Davide A1 Lee, John D A1 Leeman, Susan E A1 Leprince, Jérôme A1 Li, Xaria X A1 Williams, Tom Lloyd A1 Lolait, Stephen J A1 Lupp, Amelie A1 Macrae, Robyn A1 Maguire, Janet A1 Mazella, Jean A1 McArdle, Craig A A1 Melmed, Shlomo A1 Michel, Martin C A1 Miller, Laurence J A1 Mitolo, Vincenzo A1 Mouillac, Bernard A1 Müller, Christa E A1 Murphy, Philip A1 Nahon, Jean-Louis A1 Ngo, Tony A1 Norel, Xavier A1 Nyimanu, Duuamene A1 O'Carroll, Anne-Marie A1 Offermanns, Stefan A1 Panaro, Maria Antonietta A1 Parmentier, Marc A1 Pertwee, Roger G A1 Pin, Jean-Philippe A1 Prossnitz, Eric R A1 Quinn, Mark A1 Ramachandran, Rithwik A1 Ray, Manisha A1 Reinscheid, Rainer K A1 Rondard, Philippe A1 Rovati, G Enrico A1 Ruzza, Chiara A1 Sanger, Gareth J A1 Schöneberg, Torsten A1 Schulte, Gunnar A1 Schulz, Stefan A1 Segaloff, Deborah L A1 Serhan, Charles N A1 Stoddart, Leigh A A1 Sugimoto, Yukihiko A1 Summers, Roger A1 Tan, Valerie P A1 Thal, David A1 Thomas, Walter Wally A1 Timmermans, Pieter B M W M A1 Tirupula, Kalyan A1 Tulipano, Giovanni A1 Unal, Hamiyet A1 Unger, Thomas A1 Valant, Celine A1 Vanderheyden, Patrick A1 Vaudry, David A1 Vaudry, Hubert A1 Vilardaga, Jean-Pierre A1 Walker, Christopher S A1 Wang, Ji Ming A1 Ward, Donald T A1 Wester, Hans-Jürgen A1 Willars, Gary B A1 Woodruff, Trent M A1 Yao, Chengcan A1 Ye, Richard D AB The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (www.guidetopharmacology.org), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes over 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at http://onlinelibrary.wiley.com/doi/bph.15538. G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2021, and supersedes data presented in the 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate. YR 2021 FD 2021 LK https://hdl.handle.net/10668/25043 UL https://hdl.handle.net/10668/25043 LA en DS RISalud RD Apr 5, 2025